trpv1 antagonist
由 AP Koivisto 著作 · 2022 · 被引用 331 次 — Because TRPV1 agonists that cause desensitization can be perceived as functional antagonists of the receptor (Fig. 2), it has been postulated ... ,由 A Garami 著作 · 2010 · 被引用 198 次 — TRPV1 antagonists differentially block three modes of TRPV1 activation: by heat, protons, and chemical ligands (e.g., capsaicin). We asked what combination of ... ,The TRPV1 receptor is a ligand gated ion channel that has been implicated in mediation of many types of pain and therefore studied most extensively. The first ... ,由 J Caballero 著作 · 2022 · 被引用 13 次 — The design of TRPV1 antagonists and agonists has reached a new era since TRPV1 structures at near-atomic resolution are available. ,由 K Zhu 著作 · 2023 · 被引用 10 次 — TRPV1 antagonists treat pain and itch sensations by inhibiting receptor potential and preventing nociceptive signals from transmitting from ... ,由 MR Brandt 著作 · 2012 · 被引用 59 次 — Initial clinical results indicate that TRPV1 antagonist decrease thermal pain perception in normal subjects and elevate core body temperature [26,27,28]. ,Other potent and selective TRPV1 antagonists of both human and rat TRPV1 receptors, the 1-isoquinolin-5-yl-3-(4- trifluoromethyl-benzyl)urea, A-425619 (Abbott) ... ,由 R Brito 著作 · 2014 · 被引用 169 次 — Gadolinium blocks Ca2+-permeant, mechanosensitive cation channels and ruthenium red, a noncompetitive antagonist of TRPV1, is also a blocker of numerous cation ... ,由 T Xiao 著作 · 2023 · 被引用 21 次 — Some studies have revealed that TRPV1 antagonists have certain antidepressant and antianxiety effects, which may be beneficial to rosacea ... ,Antagonists of TRPV1 include ruthenium red, a dye that exhibits properties of noncompetitive antagonism for the TRPV1, and has a poorly defined mechanism of ...
| 相關軟體 REAPER 資訊 | |
|---|---|
 trpv1 antagonist 相關參考資料
Advances in TRP channel drug discovery: from target ...
由 AP Koivisto 著作 · 2022 · 被引用 331 次 — Because TRPV1 agonists that cause desensitization can be perceived as functional antagonists of the receptor (Fig. 2), it has been postulated ... https://www.nature.com Contributions of Different Modes of TRPV1 Activation to ...
由 A Garami 著作 · 2010 · 被引用 198 次 — TRPV1 antagonists differentially block three modes of TRPV1 activation: by heat, protons, and chemical ligands (e.g., capsaicin). We asked what combination of ... https://www.ncbi.nlm.nih.gov Discovery and development of TRPV1 antagonists
The TRPV1 receptor is a ligand gated ion channel that has been implicated in mediation of many types of pain and therefore studied most extensively. The first ... https://en.wikipedia.org Full article: A new era for the design of TRPV1 antagonists ...
由 J Caballero 著作 · 2022 · 被引用 13 次 — The design of TRPV1 antagonists and agonists has reached a new era since TRPV1 structures at near-atomic resolution are available. https://www.tandfonline.com Progress in the development of TRPV1 small-molecule ...
由 K Zhu 著作 · 2023 · 被引用 10 次 — TRPV1 antagonists treat pain and itch sensations by inhibiting receptor potential and preventing nociceptive signals from transmitting from ... https://www.sciencedirect.com TRPV1 Antagonists and Chronic Pain: Beyond Thermal ...
由 MR Brandt 著作 · 2012 · 被引用 59 次 — Initial clinical results indicate that TRPV1 antagonist decrease thermal pain perception in normal subjects and elevate core body temperature [26,27,28]. https://www.mdpi.com TRPV1 Antagonists as Analgesic Agents
Other potent and selective TRPV1 antagonists of both human and rat TRPV1 receptors, the 1-isoquinolin-5-yl-3-(4- trifluoromethyl-benzyl)urea, A-425619 (Abbott) ... https://openpainjournal.com TRPV1: A Potential Drug Target for Treating Various ...
由 R Brito 著作 · 2014 · 被引用 169 次 — Gadolinium blocks Ca2+-permeant, mechanosensitive cation channels and ruthenium red, a noncompetitive antagonist of TRPV1, is also a blocker of numerous cation ... https://www.ncbi.nlm.nih.gov TRPV1: A promising therapeutic target for skin aging and ...
由 T Xiao 著作 · 2023 · 被引用 21 次 — Some studies have revealed that TRPV1 antagonists have certain antidepressant and antianxiety effects, which may be beneficial to rosacea ... https://www.frontiersin.org Vanilloid Receptor 1 Antagonist - an overview
Antagonists of TRPV1 include ruthenium red, a dye that exhibits properties of noncompetitive antagonism for the TRPV1, and has a poorly defined mechanism of ... https://www.sciencedirect.com |